Discovery of a novel melanin concentrating hormone receptor 1 (MCHR1) antagonist with reduced hERG inhibition-Reference-Cited by-同舟云学术

Discovery of a novel melanin concentrating hormone receptor 1 (MCHR1) antagonist with reduced hERG inhibition

Published:2012-06 Issue:11 Volume:22 Page:3781-3785
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Mihalic Jeffrey T.,Fan Pingchen,Chen Xiaoqi,Chen Xi,Fu Ying,Motani Alykhan,Liang Lingming,Lindstrom Michelle,Tang Liang,Chen Jin-Long,Jaen Juan,Dai Kang,Li Leping

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference33 articles.

1. Characterization of Melanin-Concentrating Hormone from Rat Hypothalamus*

2. Structure of the Human Melanin Concentrating Hormone mRNA

3. The Rat Melanin-Concentrating Hormone Messenger Ribonucleic Acid Encodes Multiple Putative Neuropeptides Coexpressed in the Dorsolateral Hypothalamus*

4. Melanin-concentrating hormone: a functional melanocortin antagonist in the hypothalamus

5. Acute and chronic administration of melanin-concentrating hormone enhances food intake and body weight in Wistar and Sprague–Dawley rats

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