Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings-Reference-Cited by-同舟云学术

Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings

Published:2018-07 Issue:13 Volume:28 Page:2320-2323
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Willemse Tom,Eiselt Emilie,Hollanders Karlijn,Schepens Wim,van Vlijmen Herman W.T.,Chung Nga N.,Blais Véronique,Holleran Brain,Longpré Jean-Michel,Schiller Peter W.,Maes Bert U.W.,Sarret Philippe,Gendron Louis,Ballet Steven

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference35 articles.

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2. Opioid Receptors

3. Opioid Peptides: Biology, Chemistry, and Genetics: The Peptides: Analysis, Synthesis;Udenfriend,1984

4. Multitarget opioid ligands in pain relief: New players in an old game

5. The Opioid μ Agonist/δ Antagonist DIPP-NH2[Ψ] Produces a Potent Analgesic Effect, No Physical Dependence, and Less Tolerance than Morphine in Rats

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2. Endogenous Opiates and Behavior: 2018;Peptides;2020-10

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5. Corrigendum to “Chemical space screening around Phe3 in opioid peptides: Modulating µ versus δ agonism by Suzuki-Miyaura cross-couplings” [Bioorg. Med. Chem. Lett. 28(13) (2018) 2320–2323];Bioorganic & Medicinal Chemistry Letters;2018-11