Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors-Reference-Cited by-同舟云学术

Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors

Published:2016-09 Issue:17 Volume:26 Page:4216-4222
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Meegalla Sanath K.,Huang Hui,Illig Carl R.,Parks Daniel J.,Chen Jinsheng,Lee Yu-Kai,Wilson Kenneth J.,Patel Sharmila K.,Cheung Wing S.,Lu Tianbao,Kirchner Thomas,Askari Hossein B.,Geisler John,Patch Raymond J.,Gibbs Alan C.,Rady Brian,Connelly Margery,Player Mark R.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference12 articles.

1. Current Landscape of Phosphodiesterase 10A (PDE10A) Inhibition

2. K. U. Leuven Research and Development. WO2005/120474.

3. PDE-10A inhibitors as insulin secretagogues

4. Janssen Pharmaceutica NV. WO2011/051342.

5. Black S.C.; Gibbs E.M.; McNeish J.D. WO 2005/041972 2005.

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