Lead generation of 1,2-dithiolanes as exon 19 and exon 21 mutant EGFR tyrosine kinase inhibitors-Reference-Cited by-同舟云学术

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Lead generation of 1,2-dithiolanes as exon 19 and exon 21 mutant EGFR tyrosine kinase inhibitors

Published:2019-06 Issue:12 Volume:29 Page:1435-1439
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Mansour Tarek S.,Potluri Vijay,Pallepati Ranga R.,Basetti Vishnu,Keesara Mallaiah,Moghudula Ashok G.,Maiti Pranab

Funder

NCI

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. Cancer stats 2017;Siegel;CA Cancer J Clin,2017

2. Challenges and perspectives on the development of small-molecule EGFR inhibitors against T790M-mediated resistance in non-small-cell lung cancer;Song;J Med Chem,2016

3. Recent progress of small-molecule epidermal growth factor receptor (EGFR) inhibitors against C797S in non-small-cell lung cancer;Chen;J Med Chem,2018

4. Precedence and promise of covalent inhibitors of EGFR and KRAS for patients with non-small-cell lung cancer;Cheng;ACS Med Chem Lett,2018

5. Discovery of (R,E)-N-(7-Chloro-1-(1-[4-(dimethylamino)but-2-enoyl]azepan-3-yl)-1H-benzo[d]imidazol-2-yl)-2-methylisonicotinamide (EGF816), a Novel, Potent, and WT Sparing Covalent Inhibitor of Oncogenic (L858R, ex19del) and Resistant (T790M) EGFR Mutants for the Treatment of EGFR Mutant Non-Small-Cell Lung Cancers

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1. Asparagusic Acid – A Unique Approach toward Effective Cellular Uptake of Therapeutics: Application, Biological Targets, and Chemical Properties;ChemMedChem;2023-07-06

2. Regio- and stereoselective ring contraction of 1,2-dithianes to 1,2-dithiolanes;Tetrahedron Letters;2023-05

3. Dual target inhibitors based on EGFR: Promising anticancer agents for the treatment of cancers (2017-);European Journal of Medicinal Chemistry;2022-01

4. Recent contributions of quinolines to antimalarial and anticancer drug discovery research;European Journal of Medicinal Chemistry;2021-12

5. Thiol-Mediated Uptake;JACS Au;2021-05-03

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