Application of oxime-diversification to optimize ligand interactions within a cryptic pocket of the polo-like kinase 1 polo-box domain-Reference-Cited by-同舟云学术

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Application of oxime-diversification to optimize ligand interactions within a cryptic pocket of the polo-like kinase 1 polo-box domain

Published:2016-10 Issue:20 Volume:26 Page:5009-5012
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Zhao Xue Zhi,Hymel David,Burke Terrence R.

Funder

NIH Intramural Program

Center for Cancer Research, National Cancer Institute

National Institutes of Health

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. Multifaceted polo-like kinases: drug targets and antitargets for cancer therapy

2. Recent Advances and New Strategies in Targeting Plk1 for Anticancer Therapy

3. Understanding the Polo Kinase machine

4. Using Ligand-Mapping Simulations to Design a Ligand Selectively Targeting a Cryptic Surface Pocket of Polo-Like Kinase 1

5. Structural and functional analyses of minimal phosphopeptides targeting the polo-box domain of polo-like kinase 1

Cited by 18 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Affinity enhancement of polo-like kinase 1 polo box domain-binding ligands by a bivalent approach using a covalent kinase-binding component;RSC Chemical Biology;2024

2. Solid‐Phase Synthesis and Biological Evaluation of Peptides ADP‐Ribosylated at Histidine;Angewandte Chemie International Edition;2023-11-14

3. Solid‐Phase Synthesis and Biological Evaluation of Peptides ADP‐Ribosylated at Histidine;Angewandte Chemie;2023-11-14

4. Identification of multidentate tyrosyl-DNA phosphodiesterase 1 (TDP1) inhibitors that simultaneously access the DNA, protein and catalytic-binding sites by oxime diversification;RSC Chemical Biology;2023

5. Pd-catalyzed heteroannulation of isoxazoles: Convergent synthesis of isoxazolo[5,4-c]quinolines;Tetrahedron Letters;2023-01

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