Rational design of 6-methylsulfonylindoles as selective cyclooxygenase-2 inhibitors-Reference-Cited by-同舟云学术

Rational design of 6-methylsulfonylindoles as selective cyclooxygenase-2 inhibitors

Published:2004-09 Issue:18 Volume:14 Page:4741-4745
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Campbell Jeffrey A.,Bordunov Viola,Broka Chris A.,Browner Michelle F.,Kress James M.,Mirzadegan Tara,Ramesha Chakk,Sanpablo Bong F.,Stabler Russell,Takahara Patricia,Villasenor Armando,Walker Keith A.M.,Wang Jin-Hai,Welch Mary,Weller Paul

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference25 articles.

1. NS-398, a new anti-inflammatory agent, selectively inhibits prostaglandin G/H synthase/cyclooxygenase (COX-2) activity in vitro

2. Preliminary study of the safety and efficacy of SC-58635, a novel cyclooxygenase 2 inhibitor: Efficacy and safety in two placebo-controlled trials in osteoarthritis and rheumatoid arthritis, and studies of gastrointestinal and platelet effects

3. Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors: Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide (SC-58635, Celecoxib)

4. The discovery of rofecoxib, [MK 966, VIOXX®, 4-(4′-methylsulfonylphenyl)-3-phenyl-2(5H)-furanone], an orally active cyclooxygenase-2 inhibitor

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