The discovery of rofecoxib, [MK 966, VIOXX®, 4-(4′-methylsulfonylphenyl)-3-phenyl-2(5H)-furanone], an orally active cyclooxygenase-2 inhibitor-Reference-Cited by-同舟云学术

The discovery of rofecoxib, [MK 966, VIOXX®, 4-(4′-methylsulfonylphenyl)-3-phenyl-2(5H)-furanone], an orally active cyclooxygenase-2 inhibitor

Published:1999-07 Issue:13 Volume:9 Page:1773-1778
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Prasit P,Wang Z,Brideau C,Chan C.-C,Charleson S,Cromlish W,Ethier D,Evans J.F,Ford-Hutchinson A.W,Gauthier J.Y,Gordon R,Guay J,Gresser M,Kargman S,Kennedy B,Leblanc Y,Léger S,Mancini J,O'Neill G.P,Ouellet M,Percival M.D,Perrier H,Riendeau D,Rodger I,Tagari P,Thérien M,Vickers P,Wong E,Xu L.-J,Young R.N,Zamboni R,Boyce S,Rupniak N,Forrest M,Visco D,Patrick D

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. Mechanism of selective inhibition of human prostaglandin G/H synthase-1 and -2 in intact cells

2. A human whole blood assay for clinical evaluation of biochemical efficacy of cyclooxygenase inhibitors

3. The Clinical Implications of Inhibition of the Inducible Form of Cyclo-Oxygenase

4. Chapter 21. Selective Cyclooxygenase-2 Inhibitors

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