Potent and orally active non-peptide antagonists of the human melanocortin-4 receptor based on a series of trans-2-disubstituted cyclohexylpiperazines-Reference-Cited by-同舟云学术

Potent and orally active non-peptide antagonists of the human melanocortin-4 receptor based on a series of trans-2-disubstituted cyclohexylpiperazines

Published:2005-10 Issue:19 Volume:15 Page:4389-4395
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Tucci Fabio C.,White Nicole S.,Markison Stacy,Joppa Margaret,Tran Joe A.,Fleck Beth A.,Madan Ajay,Dyck Brian P.,Parker Jessica,Pontillo Joseph,Melissa Arellano L.,Marinkovic Dragan,Jiang Wanlong,Chen Caroline W.,Gogas Kathleen R.,Goodfellow Val S.,Saunders John,Foster Alan C.,Chen Chen

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference22 articles.

1. Cancer Anorexia-Cachexia Syndrome: Current Issues in Research and Management

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3. Cancer cachexia: A therapeutic approach

4. Systematic review of megestrol acetate in the treatment of anorexia-cachexia syndrome

5. New aspects on the melanocortins and their receptors

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