Synthesis and in vitro evaluation of small-molecule [18F] labeled gonadotropin-releasing hormone (GnRH) receptor antagonists as potential PET imaging agents for GnRH receptor expression-Reference-Cited by-同舟云学术

Synthesis and in vitro evaluation of small-molecule [18F] labeled gonadotropin-releasing hormone (GnRH) receptor antagonists as potential PET imaging agents for GnRH receptor expression

Published:2014-04 Issue:7 Volume:24 Page:1846-1850
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Olberg Dag Erlend,Andressen Kjetil Wessel,Levy Finn Olav,Klaveness Jo,Haraldsen Ira,Sutcliffe Julie L.

Funder

United States Department of Energy, DE-SC0002061 and in part from NIH

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. GnRH analogues—agonists and antagonists

2. Gonadotropin-releasing hormone (GnRH) and its natural analogues: A review

3. GnRH Receptors in Cancer: From Cell Biology to Novel Targeted Therapeutic Strategies

4. The Extrapituitary Effects of GnRH Antagonists and Their Potential Clinical Implications: A Narrated Review

5. Gonadotropin-releasing hormone and its receptor in normal and malignant cells

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