Identification and profiling of 3,5-dimethyl-isoxazole-4-carboxylic acid [2-methyl-4-((2S,3′S)-2-methyl-[1,3′]bipyrrolidinyl-1′-yl)phenyl] amide as histamine H3 receptor antagonist for the treatment of depression-Reference-Cited by-同舟云学术

Identification and profiling of 3,5-dimethyl-isoxazole-4-carboxylic acid [2-methyl-4-((2S,3′S)-2-methyl-[1,3′]bipyrrolidinyl-1′-yl)phenyl] amide as histamine H3 receptor antagonist for the treatment of depression

Published:2013-12 Issue:23 Volume:23 Page:6269-6273
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Gao Zhongli^ORCID,Hurst William J.,Czechtizky Werngard,Hall Daniel,Moindrot Nicolas,Nagorny Raisa,Pichat Philippe,Stefany David,Hendrix James A.,George Pascal G.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference33 articles.

1. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

2. Cloning and Functional Expression of the Human Histamine H3Receptor

3. Cloning and pharmacological characterization of the monkey histamine H3 receptor

4. Genetic and pharmacological aspects of histamine H3 receptor heterogeneity

5. A detailed autoradiographic mapping of histamine H3 receptors in rat brain areas

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