Synthesis and biological evaluation of novel thiadiazole amides as potent Cdc25B and PTP1B inhibitors-Reference-Cited by-同舟云学术

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Synthesis and biological evaluation of novel thiadiazole amides as potent Cdc25B and PTP1B inhibitors

Published:2014-09 Issue:17 Volume:24 Page:4125-4128
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Li Yingjun,Yu Yang,Jin Kun,Gao Lixin,Luo Tongchuan,Sheng Li,Shao Xin,Li Jia

Funder

National Science and Technology Major Projects

National Natural Science Foundation of China

Shanghai Commission of Science and Technology of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

1. Design and synthesis of novel bis-thiazolone derivatives as micromolar CDC25 phosphatase inhibitors: Effect of dimerisation on phosphatase inhibition

2. Development of a matrix-assisted laser desorption/ionization–mass spectrometry screening test to evidence reversible and irreversible inhibitors of CDC25 phosphatases

3. Design and synthesis of macrocyclic inhibitors of phosphatase Cdc25B

4. Structure-based virtual screening approach to identify novel classes of Cdc25B phosphatase inhibitors

5. Arylstibonic acids are potent and isoform-selective inhibitors of Cdc25a and Cdc25b phosphatases

Cited by 24 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Identification of 1,3,4-Thiadiazolyl-Containing Thiazolidine-2,4-dione Derivatives as Novel PTP1B Inhibitors with Antidiabetic Activity;Journal of Medicinal Chemistry;2024-05-09

2. New chromone derivatives bearing thiazolidine-2,4-dione moiety as potent PTP1B inhibitors: Synthesis and biological activity evaluation;Bioorganic Chemistry;2024-02

3. Facile synthesis of zinc acetate/niacin MOFs for use in wound healing;Biomedical Materials;2023-06-15

4. Exploring protein tyrosine phosphatases (PTP) and PTP-1B inhibitors in management of diabetes mellitus;Biomedicine & Pharmacotherapy;2022-09

5. Synthesis, characterization and biological evaluation of thiadiazole amide derivatives as nucleoside triphosphate diphosphohydrolases (NTPDases) inhibitors;Bioorganic Chemistry;2022-01

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