Evaluation of the cyclopentane-1,2-dione as a potential bio-isostere of the carboxylic acid functional group-Reference-Cited by-同舟云学术

Evaluation of the cyclopentane-1,2-dione as a potential bio-isostere of the carboxylic acid functional group

Published:2014-09 Issue:17 Volume:24 Page:4171-4175
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Ballatore Carlo,Gay Bryant,Huang Longchuan,Robinson Katie Herbst,James Michael J.,Trojanowski John Q.,Lee Virginia M.-Y.,Brunden Kurt R.,Smith Amos B.

Funder

NIH/NIA

NSF

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. Privileged Molecules for Protein Binding Identified from NMR-Based Screening

2. Carboxylic Acid (Bio)Isosteres in Drug Design

3. Design and Synthesis of [2-(8,9-Dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)- ethyl]phosphonic Acid (EAA-090), a Potent N-Methyl-d-aspartate Antagonist, via the Use of 3-Cyclobutene-1,2-dione as an Achiral α-Amino Acid Bioisostere

4. Synthesis of 3-Hydroxy-3-cyclobutene-1,2-dione Based Amino Acids

5. 3-hydroxy-3-cyclobutene-1,2-dione: Application of novel carboxylic acid bioisostere to an in-vivo active non-tetrazole angiotensin-II antagonist

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