3-hydroxy-3-cyclobutene-1,2-dione: Application of novel carboxylic acid bioisostere to an in-vivo active non-tetrazole angiotensin-II antagonist-Reference-Cited by-同舟云学术

3-hydroxy-3-cyclobutene-1,2-dione: Application of novel carboxylic acid bioisostere to an in-vivo active non-tetrazole angiotensin-II antagonist

Published:1993-04 Issue:4 Volume:3 Page:757-760
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Soll R.M.,Kinney W.A.,Primeau J.,Garrick L.,McCaully R.J.,Colatsky T.,Oshiro G.,Park C.H.,Hartupee D.,White V.,McCallum J.,Russo A.,Dinish J.,Wojdan A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference7 articles.

1. Chapter 27. Bioisosterism in Drug Design

2. The discovery of DuP 753, a potent, orally active nonpeptide angiotensin II receptor antagonist

3. Small-Ring Compounds. XXV. Phenylcyclobutadienoquinone and Related Compounds1

4. Nonpeptide angiotensin II receptor antagonists: the discovery of a series of N-(biphenylylmethyl)imidazoles as potent, orally active antihypertensives

5. 3-Stannylcyclobutenediones as nucleophilic cyclobutenedione equivalents. Synthesis of substituted cyclobutenediones and cyclobutenedione monoacetals and the beneficial effect of catalytic copper iodide on the Stille reaction

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