Solving time-dependent CYP3A4 inhibition for a series of indole-phenylacetic acid dual antagonists of the PGD2 receptors CRTH2 and DP-Reference-Cited by-同舟云学术

Solving time-dependent CYP3A4 inhibition for a series of indole-phenylacetic acid dual antagonists of the PGD2 receptors CRTH2 and DP

Published:2014-07 Issue:13 Volume:24 Page:2877-2880
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Johnson Michael G.,Liu Jim (Jiwen),Li An-Rong,van Lengerich Bettina,Wang Sophie,Medina Julio C.,Collins Tassie L.,Danao Jay,Seitz Lisa,Willee Angela,D’Souza Warren,Budelsky Alison L.,Fan Peter W.,Wong Simon G.W.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. CRTH2 and D-Type Prostanoid Receptor Antagonists as Novel Therapeutic Agents for Inflammatory Diseases

2. The roles of the prostaglandin D2 receptors DP1 and CRTH2 in promoting allergic responses

3. Antagonism of the prostaglandin D2 receptors DP1 and CRTH2 as an approach to treat allergic diseases

4. Recent Progress in Work on PGD2 Antagonists for Drugs Targeting Allergic Diseases

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