Pyrrolidine-pyrazole ureas as potent and selective inhibitors of 11β-hydroxysteroid-dehydrogenase type 1-Reference-Cited by-同舟云学术

Pyrrolidine-pyrazole ureas as potent and selective inhibitors of 11β-hydroxysteroid-dehydrogenase type 1

Published:2011-04 Issue:8 Volume:21 Page:2244-2251
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Venier Olivier,Pascal Cécile,Braun Alain,Namane Claudie,Mougenot Patrick,Crespin Olivier,Pacquet François,Mougenot Cécile,Monseau Catherine,Onofri Bénédicte,Dadji-Faïhun Rommel,Leger Céline,Ben-Hassine Majdi,Van-Pham Thao,Ragot Jean-Luc,Philippo Christophe,Güssregen Stefan,Engel Christian,Farjot Géraldine,Noah Lionel,Maniani Karima,Nicolaï Eric

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference41 articles.

1. 11β-Hydroxysteroid Dehydrogenase Type 1: A Tissue-Specific Regulator of Glucocorticoid Response

2. Inhibition of 11β-HSD1 as a novel treatment for the metabolic syndrome: do glucocorticoids play a role?

3. Inhibition of 11ß-hydroxysteroid dehydrogenase type 1 as a promising therapeutic target

4. 11 -Hydroxysteroid dehydrogenase type 1 knockout mice show attenuated glucocorticoid-inducible responses and resist hyperglycemia on obesity or stress

5. A Transgenic Model of Visceral Obesity and the Metabolic Syndrome

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