Discovery of dehydro-oxopiperazine acetamides as novel bradykinin B1 receptor antagonists with enhanced in vitro potency-Reference-Cited by-同舟云学术

Discovery of dehydro-oxopiperazine acetamides as novel bradykinin B1 receptor antagonists with enhanced in vitro potency

Published:2012-01 Issue:2 Volume:22 Page:1061-1067
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Qian Wenyuan,Chen Jian Jeffrey,Human Jason,Aya Toshihiro,Zhu Jiawang,Biswas Kaustav,Peterkin Tanya,Hungate Randall W.,Arik Leyla,Johnson Eileen,Kumar Gondi,Joseph Smriti,Jona Janan,Guo Hong-Xun,Wu Zufan

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference17 articles.

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3. Bradykinin B1 Receptor Antagonists as Potential Therapeutic Agents for Pain

4. Bradykinin B1 Receptor Antagonists as Novel Analgesics: A Retrospective of Selected Medicinal Chemistry Developments

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