Development of LM-41 and AF-2112, two flufenamic acid-derived TEAD inhibitors obtained through the replacement of the trifluoromethyl group by aryl rings-Reference-Cited by-同舟云学术

Development of LM-41 and AF-2112, two flufenamic acid-derived TEAD inhibitors obtained through the replacement of the trifluoromethyl group by aryl rings

Published:2023-10 Issue: Volume:95 Page:129488
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Fnaiche Ahmed,Mélin Léa^ORCID,Suárez Narjara González^ORCID,Paquin Alexis^ORCID,Vu Victoria^ORCID,Li Fengling,Allali-Hassani Abdellah,Bolotokova Albina,Allemand Frédéric,Gelin Muriel^ORCID,Cotelle Philippe^ORCID,Woo Simon,LaPlante Steven R.,Barsyte-Lovejoy Dalia,Santhakumar Vijayaratnam^ORCID,Vedadi Masoud,Guichou Jean-François^ORCID,Annabi Borhane^ORCID,Gagnon Alexandre^ORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

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