Benzodiazepine calcitonin gene-related peptide (CGRP) receptor antagonists: Optimization of the 4-substituted piperidine-Reference-Cited by-同舟云学术

Benzodiazepine calcitonin gene-related peptide (CGRP) receptor antagonists: Optimization of the 4-substituted piperidine

Published:2006-10 Issue:19 Volume:16 Page:5052-5056
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Burgey Christopher S.,Stump Craig A.,Nguyen Diem N.,Deng James Z.,Quigley Amy G.,Norton Beth R.,Bell Ian M.,Mosser Scott D.,Salvatore Christopher A.,Rutledge Ruth Z.,Kane Stefanie A.,Koblan Kenneth S.,Vacca Joseph P.,Graham Samuel L.,Williams Theresa M.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. Triptans Induce Vasoconstriction of Human Arteries and Veins from the Thoracic Wall

2. New insights into the molecular actions of serotonergic antimigraine drugs

3. New therapeutic target in primary headaches – blocking the CGRP receptor

4. CGRP-Receptor Antagonists — A Fresh Approach to Migraine Therapy?

5. Development of Human Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonists. 1. Potent and Selective Small Molecule CGRP Antagonists. 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1- piperidinyl]carbonyl]-d-tyrosyl]-l-lysyl]-4-(4-pyridinyl)piperazine: The First CGRP Antagonist for Clinical Trials in Acute Migraine

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