Synthesis and structure–activity relationship of imidazo(1,2-a)thieno(3,2-e)pyrazines as IKK-β inhibitors-Reference-Cited by-同舟云学术

Synthesis and structure–activity relationship of imidazo(1,2-a)thieno(3,2-e)pyrazines as IKK-β inhibitors

Published:2007-08 Issue:15 Volume:17 Page:4284-4289
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Belema Makonen,Bunker Amy,Nguyen Van N.,Beaulieu Francis,Ouellet Carl,Qiu Yuping,Zhang Yunhui,Martel Alain,Burke James R.,McIntyre Kim W.,Pattoli Mark A.,Daloisio Connie,Gillooly Kathleen M.,Clarke Wendy J.,Brassil Patrick J.,Zusi F. Chris,Vyas Dolatrai M.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference21 articles.

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2. Peptides Corresponding to the N and C Termini of IκB-α, -β, and -ε as Probes of the Two Catalytic Subunits of IκB Kinase, IKK-1 and IKK-2

3. NF-κB Regulation by IκB Kinase-2 in Rheumatoid Arthritis Synoviocytes

4. Transcriptional regulation via the NF-κB signaling module

5. The alternative NF-κB pathway from biochemistry to biology: Pitfalls and promises for future drug development

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