Quinolinone-based agonists of S1P1: Use of a N-scan SAR strategy to optimize in vitro and in vivo activity-Reference-Cited by-同舟云学术

Quinolinone-based agonists of S1P1: Use of a N-scan SAR strategy to optimize in vitro and in vivo activity

Published:2012-01 Issue:1 Volume:22 Page:527-531
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Pennington Lewis D.,Croghan Michael D.,Sham Kelvin K.C.,Pickrell Alexander J.,Harrington Paul E.,Frohn Michael J.,Lanman Brian A.,Reed Anthony B.,Lee Matthew R.,Xu Han,McElvain Michele,Xu Yang,Zhang Xuxia,Fiorino Michael,Horner Michelle,Morrison Henry G.,Arnett Heather A.,Fotsch Christopher,Tasker Andrew S.,Wong Min,Cee Victor J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. Sphingosine 1-Phosphate Receptor Signaling

2. CHEMOKINES, SPHINGOSINE-1-PHOSPHATE, AND CELL MIGRATION IN SECONDARY LYMPHOID ORGANS

3. Discovery of AMG 369, a Thiazolo[5,4-b]pyridine Agonist of S1P1 and S1P5

4. The alliance of sphingosine-1-phosphate and its receptors in immunity

5. Synthetic Sphingosine 1-Phosphate Receptor Modulators - Opportunities and Potential Pitfalls

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