Biphenyl/diphenyl ether renin inhibitors: Filling the S1 pocket of renin via the S3 pocket-Reference-Cited by-同舟云学术

Biphenyl/diphenyl ether renin inhibitors: Filling the S1 pocket of renin via the S3 pocket

Published:2011-08 Issue:16 Volume:21 Page:4836-4843
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Yuan Jing,Simpson Robert D.,Zhao Wei,Tice Colin M.,Xu Zhenrong,Cacatian Salvacion,Jia Lanqi,Flaherty Patrick T.,Guo Joan,Ishchenko Alexey,Wu Zhongren,McKeever Brian M.,Scott Boyd B.,Bukhtiyarov Yuri,Berbaum Jennifer,Panemangalore Reshma,Bentley Ross,Doe Christopher P.,Harrison Richard K.,McGeehan Gerard M.,Singh Suresh B.,Dillard Lawrence W.,Baldwin John J.,Claremon David A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference21 articles.

1. THE PREPARATION, PURIFICATION, AND AMINO ACID SEQUENCE OF A POLYPEPTIDE RENIN SUBSTRATE

2. Renin inhibitors

3. Aliskiren: the first renin inhibitor for clinical treatment

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