Discovery of novel bicyclic[3.3.0]proline peptidyl α-ketoamides as potent 3CL-protease inhibitors for SARS-CoV-2-Reference-Cited by-同舟云学术

Discovery of novel bicyclic[3.3.0]proline peptidyl α-ketoamides as potent 3CL-protease inhibitors for SARS-CoV-2

Published:2023-06 Issue: Volume:90 Page:129324
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Chen Xiaoxin,Li Peng,Huang Jianzhou,Yang Yaxun,Zhang Haoyu,Wang Zheng^ORCID,Zhu Zhenzhen,Wang Jingjing,Zhang Jianchen,Chen Kevin,He Haiying,Long Chaofeng,Chen Shuhui

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference21 articles.

1. Estimating excess mortality due to the COVID-19 pandemic: a systematic analysis of COVID-19-related mortality, 2020-21. Lancet Lond Engl. 2022;399(10334):1513-1536.

2. Estimating global, regional, and national daily and cumulative infections with SARS-CoV-2 through Nov 14, 2021: a statistical analysis. Lancet Lond Engl. 2022;399(10344):2351-2380.

3. Antiviral pills could change pandemic’s course;Couzin-Frankel;Science,2021

4. Discovery and Synthesis of a Phosphoramidate Prodrug of a Pyrrolo[2,1-f][triazin-4-amino] Adenine C-Nucleoside (GS-5734) for the Treatment of Ebola and Emerging Viruses;Siegel;J Med Chem,2017

5. An Overview of Severe Acute Respiratory Syndrome-Coronavirus (SARS-CoV) 3CL Protease Inhibitors: Peptidomimetics and Small Molecule Chemotherapy;Pillaiyar;J Med Chem,2016

Cited by 3 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis of Gem-Dimethyl Bicyclic [3.1.0] Proline as an Antiviral Drug Intermediate;Mini-Reviews in Organic Chemistry;2024-04-29

2. On the origins of SARS-CoV-2 main protease inhibitors;RSC Medicinal Chemistry;2024

3. Small-molecule anti-COVID-19 drugs and a focus on China’s homegrown mindeudesivir (VV116);Frontiers of Medicine;2023-12