Rational design of potent GSK3β inhibitors with selectivity for Cdk1 and Cdk2-Reference-Cited by-同舟云学术

Rational design of potent GSK3β inhibitors with selectivity for Cdk1 and Cdk2

Published:2010-03 Issue:6 Volume:20 Page:1985-1989
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Lesuisse Dominique,Dutruc-Rosset Gilles,Tiraboschi Gilles,Dreyer Matthias K.,Maignan Sébastien,Chevalier Alain,Halley Frank,Bertrand Philippe,Burgevin Marie-Claude,Quarteronet Dominique,Rooney Thomas

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. Phosphorylation of human tau protein by microtubule-associated kinases: GSK3? and cdk5 are key participants

2. Advances in tau-focused drug discovery for Alzheimer's disease and related tauopathies

3. The Molecular Bases of Alzheimer's Disease and Other Neurodegenerative Disorders

4. Crystal structure of cyclin-dependent kinase 2

5. Elucidation of Characteristic Structural Features of Ligand Binding Sites of Protein Kinases: A Neural Network Approach

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