Serendipitous discovery of aryl boronic acids as β-lactamase inhibitors
Author:
Funder
Merck
Publisher
Elsevier BV
Subject
Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry
Reference18 articles.
1. β-lactams and β-lactamase inhibitors: an overview;Bush;Cold Spring Harb Perspect Med,2016
2. Unmet Medical Need in Infectious Diseases
3. beta-Lactamases in laboratory and clinical resistance
4. Updated Functional Classification of β-Lactamases
5. Understanding the longevity of the β-lactam antibiotics and of antibiotic/β-lactamase inhibitor combinations
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2. Class C β-Lactamases: Molecular Characteristics;Clinical Microbiology Reviews;2022-09-21
3. The serendipitous integration of small boron-embedded molecules into medicinal chemistry;Fundamentals and Applications of Boron Chemistry;2022
4. Boronic Acids and Their Derivatives in Medicinal Chemistry: Synthesis and Biological Applications;Molecules;2020-09-21
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