Discovery and optimization of covalent EGFR T790M/L858R mutant inhibitors-Reference-Cited by-同舟云学术

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Discovery and optimization of covalent EGFR T790M/L858R mutant inhibitors

Published:2021-11 Issue: Volume:52 Page:128406
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Hoogenboom Niels,Demont Dennis,de Zwart Edwin,Verkaik Saskia,Emmelot Maaike,van de Kar Bas,Kaptein Allard,Barf Tjeerd

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference12 articles.

1. Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitor–Resistant Disease

2. Rational, biologically based treatment of EGFR-mutant non-small-cell lung cancer

3. Gefitinib or Chemotherapy for Non–Small-Cell Lung Cancer with Mutated EGFR

4. EGFRMutation and Resistance of Non–Small-Cell Lung Cancer to Gefitinib

5. Target Binding Properties and Cellular Activity of Afatinib (BIBW 2992), an Irreversible ErbB Family Blocker

Cited by 3 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Design, preparation and biological evaluation of new Rociletinib-inspired analogs as irreversible EGFR inhibitors to treat non-small-cell-lung cancer;Bioorganic & Medicinal Chemistry;2024-09

2. Identification of the Brucea javanica Constituent Brusatol as a EGFR-Tyrosine Kinase Inhibitor in a Cell-Free Assay;ACS Omega;2023-07-28

3. Development and validation of an LC-MS/MS method for simultaneous determination of SH-1028, an irreversible third-generation EGFR TKI, and two of its metabolites in human plasma: application in clinical pharmacokinetics;Xenobiotica;2023-02-01

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