Synthesis and multiparametric evaluation of thiadiazoles and oxadiazoles as diacylglycerol acyltransferase type 1 inhibitors-Reference-Cited by-同舟云学术

Synthesis and multiparametric evaluation of thiadiazoles and oxadiazoles as diacylglycerol acyltransferase type 1 inhibitors

Published:2016-01 Issue:1 Volume:26 Page:25-32
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Mougenot Patrick,Namane Claudie,Fett Eykmar,Goumy Florence,Dadji-Faïhun Rommel,Langot Gwladys,Monseau Catherine,Onofri Bénédicte,Pacquet François,Pascal Cécile,Crespin Olivier,Ben-Hassine Majdi,Ragot Jean-Luc,Van-Pham Thao,Philippo Christophe,Chatelain-Egger Florence,Péron Philippe,Le Bail Jean-Christophe,Guillot Etienne,Chamiot-Clerc Philippe,Chabanaud Marie-Aude,Pruniaux Marie-Pierre,Ménegotto Jérôme,Schmidt Friedemann,Venier Olivier,Viviani Fabrice,Nicolai Eric

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference29 articles.

1. Identification of a gene encoding an acyl CoA:diacylglycerol acyltransferase, a key enzyme in triacylglycerol synthesis

2. Sturley, S. L.; Oelkers, P. U.S. Pat. 6,100,077.

3. Cloning of DGAT2, a Second Mammalian Diacylglycerol Acyltransferase, and Related Family Members

4. Current Status of the Research and Development of Diacylglycerol O-Acyltransferase 1 (DGAT1) Inhibitors

5. New Chemical Entities Entering Phase III Trials in 2012

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