Identification of a selective inhibitor of murine intestinal alkaline phosphatase (ML260) by concurrent ultra-high throughput screening against human and mouse isozymes-Reference-Cited by-同舟云学术

Identification of a selective inhibitor of murine intestinal alkaline phosphatase (ML260) by concurrent ultra-high throughput screening against human and mouse isozymes

Published:2014-02 Issue:3 Volume:24 Page:1000-1004
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Ardecky Robert J.,Bobkova Ekaterina V.,Kiffer-Moreira Tina,Brown Brock,Ganji Santhi,Zou Jiwen,Pass Ian,Narisawa Sonoko,Iano Flávia Godoy,Rosenstein Craig,Cheltsov Anton,Rascon Justin,Hedrick Michael,Gasior Carlton,Forster Anita,Shi Shenghua,Dahl Russell,Vasile Stefan,Su Ying,Sergienko Eduard,Chung Thomas D.Y.,Kaunitz Jonathan,Hoylaerts Marc F.,Pinkerton Anthony B.,Millán José Luis

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. Mammalian Alkaline Phosphatases: From Biology to Applications in Medicine and Biotechnology;Millán,2006

2. A novel phosphatase upregulated inAkp3knockout mice

3. Disruption of the murine intestinal alkaline phosphatase geneAkp3impairs lipid transcytosis and induces visceral fat accumulation and hepatic steatosis

4. Intestinal alkaline phosphatase is a gut mucosal defense factor maintained by enteral nutrition

5. A Role for Intestinal Alkaline Phosphatase in the Maintenance of Local Gut Immunity

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