[11C-carbonyl]CEP-32496: Radiosynthesis, biodistribution and PET study of brain uptake in P-gp/BCRP knockout mice-Reference-Cited by-同舟云学术

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[11C-carbonyl]CEP-32496: Radiosynthesis, biodistribution and PET study of brain uptake in P-gp/BCRP knockout mice

Published:2014-08 Issue:15 Volume:24 Page:3574-3577
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Shimoda Yoko,Yui Joji,Fujinaga Masayuki,Xie Lin,Kumata Katsushi,Ogawa Masanao,Yamasaki Tomoteru,Hatori Akiko,Kawamura Kazunori,Zhang Ming-Rong

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference24 articles.

1. Mutations of the BRAF gene in human cancer

2. Clinicopathologic significance ofBRAF V600E mutation in papillary carcinomas of the thyroid

3. Identification of 1-(3-(6,7-Dimethoxyquinazolin-4-yloxy)phenyl)-3-(5-(1,1,1-trifluoro-2-methylpropan-2-yl)isoxazol-3-yl)urea Hydrochloride (CEP-32496), a Highly Potent and Orally Efficacious Inhibitor of V-RAF Murine Sarcoma Viral Oncogene Homologue B1 (BRAF) V600E

4. CEP-32496: A Novel Orally Active BRAFV600E Inhibitor with Selective Cellular and In Vivo Antitumor Activity

5. Tyrosine Kinase Inhibitor Gefitinib Enhances Topotecan Penetration of Gliomas

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1. Strategies for designing novel positron emission tomography (PET) radiotracers to cross the blood–brain barrier;Journal of Labelled Compounds and Radiopharmaceuticals;2023-04-14

2. [11C]phosgene: Synthesis and application for development of PET radiotracers;Nuclear Medicine and Biology;2021-01

3. Synthesis of a 11C-Isotopologue of the B-Raf-Selective Inhibitor Encorafenib Using In-Loop [11C]CO2 Fixation;ACS Omega;2020-08-16

4. Molecular imaging of membrane drug efflux transporters activity in cancer;Drug Efflux Pumps in Cancer Resistance Pathways: From Molecular Recognition and Characterization to Possible Inhibition Strategies in Chemotherapy;2020

5. Small Molecule Chemosensitizing Agents: Polo-Like Kinase 1 (Plk1), BRAF and Janus Kinase (JAK) Inhibitors;Protein Kinase Inhibitors as Sensitizing Agents for Chemotherapy;2019

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