Discovery of a potent, orally available furopyridine derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitor-Reference-Cited by-同舟云学术

Discovery of a potent, orally available furopyridine derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitor

Published:2024-09 Issue: Volume:109 Page:129848
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Hagihara Shuichi,Ishizawa Kouhei,Kikuchi Manami,Kawano Yuko,Nishidate Akiko,Matsumoto Fumi,Hashimoto Naohiro,Sasaki Chiduko,Miyaguchi Ikuko,Okada Okimasa,Akashi Tomoya,Nakayama Shinji,Ogasawara Yuko,Endo Junichi^ORCID

Publisher

Elsevier BV

Reference16 articles.

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3. A Mammalian bromodomain protein, brd4, interacts with replication factor C and inhibits progression to S phase;Maruyama;Mol Cell Biol,2002

4. Growth and early postimplantation defects in mice deficient for the bromodomain-containing protein Brd4;Houzelstein;Mol Cell Biol,2002

5. The double bromodomain protein Brd4 binds to acetylated chromatin during interphase and mitosis;Dey;Proc Natl Acad Sci USA,2003

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1. Discovery of a potent orally available pyrazolopyridone derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitor;Bioorganic & Medicinal Chemistry Letters;2024-09