Discovery of a potent orally available pyrazolopyridone derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitor
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Published:2024-09
Issue:
Volume:109
Page:129849
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ISSN:0960-894X
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Container-title:Bioorganic & Medicinal Chemistry Letters
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language:en
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Short-container-title:Bioorganic & Medicinal Chemistry Letters
Author:
Hagihara Shuichi,
Ishizawa KouheiORCID,
Soga Kana,
Honjo Takashi,
Takai Shigeki,
Kawano Yuko,
Kikuchi Manami,
Nishidate Akiko,
Matsumoto Fumi,
Murase Mikako,
Hashimoto Naohiro,
Sasaki Chiduko,
Miyaguchi Ikuko,
Okada Okimasa,
Akashi Tomoya,
Nakayama Shinji,
Ogasawara Yuko,
Endo JunichiORCID