N-substituted bis-C-alkyloxadiazolones as dual effectors: Efficient intermediates to amidoximes or amidines and prodrug candidates of potent antimalarials-Reference-Cited by-同舟云学术

N-substituted bis-C-alkyloxadiazolones as dual effectors: Efficient intermediates to amidoximes or amidines and prodrug candidates of potent antimalarials

Published:2009-09 Issue:17 Volume:19 Page:5233-5236
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Degardin Mélissa,Wein Sharon,Durand Thierry,Escale Roger,Vial Henry,Vo-Hoang Yen

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference33 articles.

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3. Potent Antimalarial Activity of 2-Aminopyridinium Salts, Amidines, and Guanidines

4. Prodrugs of bisthiazolium salts are orally potent antimalarials

5. Antimalarial Activity of Compounds Interfering with Plasmodium falciparum Phospholipid Metabolism: Comparison between Mono- and Bisquaternary Ammonium Salts

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