Phosphodiesterase type IV (PDE IV) inhibition. Synthesis and evaluation of a series of 1,3,4-trisubstituted pyrrolidines-Reference-Cited by-同舟云学术

Phosphodiesterase type IV (PDE IV) inhibition. Synthesis and evaluation of a series of 1,3,4-trisubstituted pyrrolidines

Published:1995-09 Issue:17 Volume:5 Page:1977-1982
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Stafford Jeffrey A,Valvano Nicole L,Feldman Paul L,Sloan Brawley E,Cowan David J,Domanico Paul L,Leesnitzer Michael A,Rose Dudley A,Stimpson Stephen A,Strickland Alan B,Unwalla Rayomand J,Verghese Margrith W

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference24 articles.

1. Primary sequence of cyclic nucleotide phosphodiesterase isozymes and the design of selective inhibitors

2. Differential modulation of tissue function and therapeutic potential of selective inhibitors of cyclic nucleotide phosphodiesterase isoenzymes

3. Substance P antagonists

4. Human Monocytes;Verghese,1989

5. Chapter 19. Isozyme-Selective Phosphodiesterase Inhibitors as Antiasthmatic Agents

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