Allosteric modulation of GPCRs: From structural insights to in silico drug discovery
Author:
Funder
COST
German Research Foundation
LOEWE
Publisher
Elsevier BV
Subject
Pharmacology (medical),Pharmacology
Reference140 articles.
1. The concise guide to pharmacology 2019/20: G protein-coupled receptors;Alexander;British Journal of Pharmacology,2019
2. Retrospective ensemble docking of allosteric modulators in an adenosine G-protein-coupled receptor;Bhattarai;Biochimica et Biophysica Acta (BBA) - General Subjects,2020
3. Integrated in silico fragment-based drug design: case study with allosteric modulators on metabotropic glutamate receptor 5;Bian;The AAPS Journal,2017
4. Allosteric coupling and biased agonism in G protein-coupled receptors;Bock;FEBS Journal,2021
5. Allosteric modulators targeting CNS muscarinic receptors;Bock;Neuropharmacology,2018
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