Allosteric modulators of rhodopsin-like G protein-coupled receptors: Opportunities in drug development
Author:
Publisher
Elsevier BV
Subject
Pharmacology (medical),Pharmacology
Reference185 articles.
1. MK-0677 (ibutamoren mesylate) for the treatment of patients recovering from hip fracture: a multicenter, randomized, placebo-controlled phase IIb study;Adunsky;Arch Gerontol Geriatr,2011
2. Allosteric modulator ORG27569 induces a CB1 cannabinoid receptor high affinity agonist binding state, receptor internalization and Gi-independent ERK1/2 activation;Ahn;J Biol Chem,2012
3. Interaction of the active metabolite of prasugrel, R-138727, with cysteine 97 and cysteine 175 of the human P2Y12 receptor;Algaier;J Thromb Haemost,2008
4. 2-Arylpropionic CXC chemokine receptor 1 (CXCR1) ligands as novel noncompetitive CXCL8 inhibitors;Allegretti;J Med Chem,2005
5. In vitro pharmacological characterization of RXFP3 allosterism: an example of probe dependency;Alvarez-Jaimes;PLoS One,2012
Cited by 60 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Opportunities and challenges in drug discovery targeting the orphan receptor GPR12;Drug Discovery Today;2023-09
2. In VitroBiology: Measuring Pharmacological Activity that Will Translate to Clinical Efficacy;The Handbook of Medicinal Chemistry;2023-02-03
3. Identification and characterization of select oxysterols as ligands for GPR17;British Journal of Pharmacology;2022-11-14
4. Purinergic receptors modulators: An emerging pharmacological tool for disease management;Medicinal Research Reviews;2022-05-13
5. International Union of Basic and Clinical Pharmacology. CXII: Adenosine Receptors: A Further Update;Pharmacological Reviews;2022-03-17
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3