Identification and characterization of select oxysterols as ligands for GPR17
Author:
Affiliation:
1. Janssen Research & Development, LLC San Diego California USA
Publisher
Wiley
Subject
Pharmacology
Link
https://onlinelibrary.wiley.com/doi/pdf/10.1111/bph.15969
Reference73 articles.
1. THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein‐coupled receptors
2. 3-(2-Carboxyethyl)indole-2-carboxylic Acid Derivatives: Structural Requirements and Properties of Potent Agonists of the Orphan G Protein-Coupled Receptor GPR17
3. Functional expression of opioid receptors and other human GPCRs in yeast engineered to produce human sterols
4. Distinct expression and ligand-binding profiles of two constitutively active GPR17 splice variants
5. Cholesterol-24S-hydroxylase (CYP46A1) Is Specifically Expressed in Neurons of the Neural Retina
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1. Unbiased insights into the multiplicity of the CYP46A1 brain effects in 5XFAD mice treated with low dose-efavirenz;Journal of Lipid Research;2024-06
2. Knockdown and inhibition of hippocampal GPR17 attenuates lipopolysaccharide-induced cognitive impairment in mice;Journal of Neuroinflammation;2023-11-21
3. Structural analysis of human G‐protein‐coupled receptor 17 ligand binding sites;Journal of Cellular Biochemistry;2023-02-15
4. Commentary on ‘Identification and characterization of select oxysterols as ligands for GPR17’;British Journal of Pharmacology;2023-01-20
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