Design, synthesis and biological evaluation of dihydroquinoxalinone derivatives as BRD4 inhibitors-Reference-Cited by-同舟云学术

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Design, synthesis and biological evaluation of dihydroquinoxalinone derivatives as BRD4 inhibitors

Published:2016-10 Issue: Volume:68 Page:236-244
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Yang Yifei,Zhao Leilei,Xu Bin,Yang LingYun,Zhang Jian,Zhang Huibin,Zhou Jinpei

Funder

Natural Science Foundation of Jiangsu Province

China National Key Hi-Tech Innovation Project for the R&D of Novel Drugs

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference54 articles.

1. Discovery of Epigenetic Regulator I-BET762: Lead Optimization to Afford a Clinical Candidate Inhibitor of the BET Bromodomains

2. Histone H4 acetylation and the epigenetic reader Brd4 are critical regulators of pluripotency in embryonic stem cells

3. Discovery of Benzotriazolo[4,3-d][1,4]diazepines as Orally Active Inhibitors of BET Bromodomains

4. Progress in the Development and Application of Small Molecule Inhibitors of Bromodomain–Acetyl-lysine Interactions

5. BET inhibition as a single or combined therapeutic approach in primary paediatric B-precursor acute lymphoblastic leukaemia

Cited by 25 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Direct C–H alkylation of 3,4-dihydroquinoxaline-2-ones with N-(acyloxy)phthalimides via radical–radical cross coupling;Chemical Communications;2024

2. Access to enantioenriched dihydroquinoxalinones via Cu-catalyzed propargylic substitution;Organic Chemistry Frontiers;2024

3. Catalytic Nucleophilic and Electrophilic Functionalization of Dihydroquinoxalin‐2‐ones;ChemCatChem;2023-05-09

4. Photocatalytic Functionalization of Dihydroquinoxalin‐2‐Ones with Pyrazolones;Advanced Synthesis & Catalysis;2022-11-21

5. Chemoenzymatic Asymmetric Synthesis of Complex Heterocycles: Dihydrobenzoxazinones and Dihydroquinoxalinones;ACS Catalysis;2022-09-06

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