Simple heteroaryl modifications in the 4,5-diarylisoxazol-3-carboxylic acid scaffold favorably modulates the activity as dual mPGES-1/5-LO inhibitors with in vivo efficacy-Reference-Cited by-同舟云学术

Simple heteroaryl modifications in the 4,5-diarylisoxazol-3-carboxylic acid scaffold favorably modulates the activity as dual mPGES-1/5-LO inhibitors with in vivo efficacy

Published:2021-07 Issue: Volume:112 Page:104861
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Gürses Tuğba,Olğaç Abdurrahman,Garscha Ulrike,Gür Maz Tuğçe,Bal Nur Banu,Uludağ Orhan,Çalışkan Burcu,Schubert Ulrich S.,Werz Oliver,Banoglu Erden

Funder

Turkish Academy of Sciences

Deutsche Forschungsgemeinschaft

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

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