Chemical space exploration of novel naphthyl-carboxamide-diarylpyrimidine derivatives with potent anti-HIV-1 activity-Reference-Cited by-同舟云学术

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Chemical space exploration of novel naphthyl-carboxamide-diarylpyrimidine derivatives with potent anti-HIV-1 activity

Published:2021-06 Issue: Volume:111 Page:104905
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Sang Yali,Pannecouque Christophe,De Clercq Erik,Zhuang Chunlin,Chen Fener

Funder

Fudan University

National Natural Science Foundation of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference21 articles.

1. Development of non-nucleoside reverse transcriptase inhibitors (NNRTIs): our past twenty years;Zhuang;Acta Pharm. Sin. B,2020

2. Structural modifications of DAPY analogues with potent anti-HIV-1 activity;Feng;ChemMedChem,2009

3. Fragment-based discovery of sulfur-containing diarylbenzopyrimidines as novel nonnucleoside reverse transcriptase inhibitors;Han;Chin. Chem. Lett.,2020

4. Molecular Hybridization-Inspired Optimization of Diarylbenzopyrimidines as HIV-1 Nonnucleoside Reverse Transcriptase Inhibitors with Improved Activity against K103N and E138K Mutants and Pharmacokinetic Profiles;Han;ACS Infect. Dis.,2020

5. Design and synthesis of conformationally constrained inhibitors of non-nucleoside reverse transcriptase;Gomez;J. Med. Chem.,2011

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Structure-based discovery of novel piperidine-biphenyl-DAPY derivatives as non-nucleoside reverse transcriptase inhibitors featuring improved potency, safety, and selectivity: From piperazine-biphenyl-DAPYs to piperidine-biphenyl-DAPYs;European Journal of Medicinal Chemistry;2024-10

2. Deciphering the enigmas of non‐nucleoside reverse transcriptase inhibitors (NNRTIs): A medicinal chemistry expedition towards combating HIV drug resistance;Medicinal Research Reviews;2024-08-26

3. Picomolar inhibitor of reverse transcriptase featuring significantly improved metabolic stability;Acta Pharmaceutica Sinica B;2023-07

4. Fragment Hopping-Based Design of Novel Biphenyl-DAPY Derivatives as Potent Non-Nucleoside Reverse Transcriptase Inhibitors Featuring Significantly Improved Anti-Resistance Efficacy;Journal of Medicinal Chemistry;2023-03-30

5. Diarylpyrimidines and related analogs as antiviral agents;Privileged Scaffolds in Drug Discovery;2023

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