Design and Synthesis of Conformationally Constrained Inhibitors of Non-Nucleoside Reverse Transcriptase-Reference-Cited by-同舟云学术

Design and Synthesis of Conformationally Constrained Inhibitors of Non-Nucleoside Reverse Transcriptase

Published:2011-10-28 Issue:22 Volume:54 Page:7920-7933
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gomez Robert¹,Jolly Samson J.¹,Williams Theresa¹,Vacca Joseph P.¹,Torrent Maricel¹,McGaughey Georgia¹,Lai Ming-Tain¹,Felock Peter¹,Munshi Vandna¹,DiStefano Daniel¹,Flynn Jessica¹,Miller Mike¹,Yan Youwei¹,Reid John¹,Sanchez Rosa¹,Liang Yuexia¹,Paton Brenda¹,Wan Bang-Lin¹,Anthony Neville¹

Affiliation:

1. Departments of †West Point Discovery Chemistry, ‡Chemistry Modeling and Informatics, §In Vitro Pharmacology, ∥Vaccine Research, ⊥ID Antiviral HIV Discovery, #Structural Chemistry, and ∞DMPK Preclinical WP, Merck Research Labs., 770 Sumneytown Pike, P.O. Box 4, West Point, Pennsylvania 19486-0004, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm2010173

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