Novel N-substituted 5-phosphate-d-arabinonamide derivatives as strong inhibitors of phosphoglucose isomerases: Synthesis, structure-activity relationship and crystallographic studies-Reference-Cited by-同舟云学术

Novel N-substituted 5-phosphate-d-arabinonamide derivatives as strong inhibitors of phosphoglucose isomerases: Synthesis, structure-activity relationship and crystallographic studies

Published:2020-09 Issue: Volume:102 Page:104048
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Ahmad Lama,Plancqueel Stéphane,Lazar Noureddine,Korri-Youssoufi Hafsa,Li de la Sierra-Gallay Inès,van Tilbeurgh Herman,Salmon Laurent

Funder

French Infrastructure for Integrated Structural Biology

Laboratoire d'Excellence en Recherche sur le Médicament et l'Innovation Thérapeutique

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference45 articles.

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3. Synthesis and evaluation of a new inhibitor of phosphoglucose isomerase: the enediolate analogue 5-phospho-D-arabinohydroxamate;Hardré;Bioorg. Med. Chem. Lett.,1998

4. The enediolate analogue 5-phosphoarabinonate as a mechanistic probe for phosphoglucose isomerase;Chirgwin;J. Biol. Chem.,1975

5. The crystal structure of human phosphoglucose isomerase at 1.6 A resolution: implications for catalytic mechanism, cytokine activity and haemolytic anaemia;Read;J. Mol. Biol.,2001

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