Discovery of novel quinolin-2-one derivatives as potential GSK-3β inhibitors for treatment of Alzheimer’s disease: Pharmacophore-based design, preliminary SAR, in vitro and in vivo biological evaluation-Reference-Cited by-同舟云学术

Discovery of novel quinolin-2-one derivatives as potential GSK-3β inhibitors for treatment of Alzheimer’s disease: Pharmacophore-based design, preliminary SAR, in vitro and in vivo biological evaluation

Published:2024-05 Issue: Volume:146 Page:107324
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Abdo Moustafa Esraa,Abdelrasheed Allam Heba,Fouad Marwa A.,El Kerdawy Ahmed M.,Nasser Eid El-Sayed Nahed,Wagner Christoph,Abdel-Aziz Hatem A.,Abdel Fattah Ezzat Manal

Publisher

Elsevier BV

Reference65 articles.

1. Recent advances in the neurobiology and neuropharmacology of Alzheimer's disease;Kumar;Biomed. Pharmacother.,2018

2. The worldwide economic impact of dementia 2010;Wimo;Alzheimer's Dement.,2013

3. Design, synthesis, in vitro, and in vivo evaluation of novel phthalazinone-based derivatives as promising acetylcholinesterase inhibitors for treatment of Alzheimer's disease;Ezzat;Drug Dev. Res.,2023

4. A comprehensive description of GluN2B-selective N-methyl-D-aspartate (NMDA) receptor antagonists;Liu;Eur. J. Med. Chem.,2020

5. New pharmacological strategies for treatment of Alzheimer's disease: focus on disease modifying drugs;Salomone;Br. J. Clin. Pharmacol.,2012

Cited by 2 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Metal‐Free Photocyclization/Oxidation Cascade Constructing Quinoline‐2‐ones and Tetrahydrocarbazolones;Advanced Synthesis & Catalysis;2024-09-05

2. Design, synthesis, antineoplastic activity of new pyrazolo[3,4-d]pyrimidine derivatives as dual CDK2/GSK3β kinase inhibitors; molecular docking study, and ADME prediction;Bioorganic Chemistry;2024-09