Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic h CA II and membrane-bound h CA IX isoforms-Reference-Cited by-同舟云学术

Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic h CA II and membrane-bound h CA IX isoforms

Published:2018-02 Issue: Volume:76 Page:88-97
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Krasavin Mikhail,Shetnev Anton,Sharonova Tatyana,Baykov Sergey^ORCID,Tuccinardi Tiziano,Kalinin Stanislav,Angeli Andrea,Supuran Claudiu T.

Funder

Russian Scientific Fund

Russian Federation Ministry of Education and Science

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference41 articles.

1. Multiple binding modes of inhibitors to carbonic anhydrases: how to design specific drugs targeting 15 different isoforms?;Alterio;Chem. Rev.,2012

2. Diuretics: from classical carbonic anhydrase inhibitors to novel applications of the sulfonamides;Supuran;Curr. Pharm. Des.,2008

3. The development of topically acting carbonic anhydrase inhibitors as antiglaucoma agents;Supuran;Curr. Pharm. Des.,2008

4. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators;Supuran;Nat. Rev. Drug Discov.,2008

5. Carbonic anhydrase inhibitors and activators for novel therapeutic applications;Supuran;Future Med. Chem.,2011

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