Characterisation of utrophin modulator SMT C1100 as a non-competitive inhibitor of firefly luciferase-Reference-Cited by-同舟云学术

Characterisation of utrophin modulator SMT C1100 as a non-competitive inhibitor of firefly luciferase

Published:2020-01 Issue: Volume:94 Page:103395
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Wilkinson Isabel V.L.,Reynolds Jessica K.,Galan Sébastien R.G.,Vuorinen Aini,Sills Adam J.,Pires Elisabete,Wynne Graham M.,Wilson Francis X.,Russell Angela J.

Funder

Engineering and Physical Sciences Research Council

Medical Research Council

Muscular Dystrophy UK

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference63 articles.

1. Illuminating insights into firefly luciferase and other bioluminescent reporters used in chemical biology;Thorne;Chem. Biol.,2010

2. Bioluminescent assays for high-throughput screening;Fan;Assay Drug Dev. Technol.,2007

3. Modulation of firefly luciferase stability and impact on studies of gene regulation;Thompson;Gene,1991

4. Firefly luciferase in chemical biology: A compendium of inhibitors, mechanistic evaluation of chemotypes, and suggested use as a reporter;Thorne;Chem. Biol.,2012

5. Profile of the GSK published protein kinase inhibitor set across ATP-dependent and-independent luciferases: implications for reporter-gene assays;Dranchak;PLoS ONE,2013

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