Synthesis of aryl pyrazole via Suzuki coupling reaction, in vitro mushroom tyrosinase enzyme inhibition assay and in silico comparative molecular docking analysis with Kojic acid-Reference-Cited by-同舟云学术

Synthesis of aryl pyrazole via Suzuki coupling reaction, in vitro mushroom tyrosinase enzyme inhibition assay and in silico comparative molecular docking analysis with Kojic acid

Published:2018-09 Issue: Volume:79 Page:293-300
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Channar Pervaiz Ali,Saeed Aamer,Larik Fayaz Ali,Batool Bakhtawar,Kalsoom Saima,Hasan M.M,Erben Mauricio F.,El-Seedi Hesham R.,Ali Musrat,Ashraf Zaman

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference30 articles.

1. Synthesis and biological evaluation of novel hydroxybenzaldehyde-based kojic acid analogues as inhibitors of mushroom tyrosinase

2. Carvacrol derivatives as mushroom tyrosinase inhibitors; synthesis, kinetics mechanism and molecular docking studies

3. Inhibitory effects of 4-chlorocinnamaldehyde on the activity of mushroom tyrosinase

4. Structural insight into the active site of mushroom tyrosinase using phenylbenzoic acid derivatives

5. Chemical exploration of 4-(4-fluorobenzyl)piperidine fragment for the development of new tyrosinase inhibitors

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