The solubility, permeability and the dose as key factors in formulation development for oral lipophilic drugs: Maximizing the bioavailability of carbamazepine with a cosolvent-based formulation-Reference-Cited by-同舟云学术

The solubility, permeability and the dose as key factors in formulation development for oral lipophilic drugs: Maximizing the bioavailability of carbamazepine with a cosolvent-based formulation

Published:2020-05 Issue: Volume:582 Page:119307
ISSN:0378-5173
Container-title:International Journal of Pharmaceutics
language:en
Short-container-title:International Journal of Pharmaceutics

Author:

Fine-Shamir Noa,Beig Avital,Miller Jonathan M.,Dahan Arik

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference39 articles.

1. Theoretical and experimental studies of transport of micelle-solubilized solutes;Amidon;J. Pharm. Sci.,1982

2. Oral delivery of lipophilic drugs: the tradeoff between solubility increase and permeability decrease when using cyclodextrin-based formulations;Beig;PLoS One,2013

3. Quantification of carbamazepine and its 10,11-epoxide metabolite in rat plasma by UPLC-UV and application to pharmacokinetic study;Beig;Biomed. Chromatogr.,2014

4. Advantageous solubility-permeability interplay when using amorphous solid dispersion (ASD) formulation for the BCS Class IV P-gp substrate Rifaximin: simultaneous increase of both the solubility and the permeability;Beig;AAPS J.,2017

5. Concomitant solubility-permeability increase: Vitamin E TPGS vs. amorphous solid dispersion as oral delivery systems for etoposide;Beig;Eur. J. Pharm. Biopharm.,2017

Cited by 15 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Formulation of semi-solid dosage forms indented for transdermal delivery of ivermectin;Journal of Drug Delivery Science and Technology;2024-09

2. Preparation, Optimization, and Anti-Pulmonary Infection Activity of Casein-Based Chrysin Nanoparticles;International Journal of Nanomedicine;2024-06

3. Ethanol-based solubility-enabling oral drug formulation development: Accounting for the solubility-permeability interplay;International Journal of Pharmaceutics;2024-03

4. From waste to a resource? Hemicelluloses enhance the dissolution and stability of the amorphous state of carbamazepine;Sustainable Chemistry and Pharmacy;2024-02

5. Mechanistic Insight in Permeability through Different Membranes in the Presence of Pharmaceutical Excipients: A Case of Model Hydrophobic Carbamazepine;Pharmaceutics;2024-01-28