Oral Delivery of Lipophilic Drugs: The Tradeoff between Solubility Increase and Permeability Decrease When Using Cyclodextrin-Based Formulations
Author:
Publisher
Public Library of Science (PLoS)
Subject
Multidisciplinary
Reference40 articles.
1. Rationalizing the selection of oral lipid based drug delivery systems by an in vitro dynamic lipolysis model for improved oral bioavailability of poorly water soluble drugs;A Dahan;Journal of Controlled Release,2008
2. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings;CA Lipinski;Advanced Drug Delivery Reviews,2001
3. A theoretical basis for a biopharmaceutic drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability;GL Amidon;Pharmaceutical Research,1995
4. Prediction of solubility and permeability class membership: Provisional BCS classification of the world’s top oral drugs;A Dahan;The AAPS Journal,2009
5. High-permeability criterion for BCS classification: Segmental/pH dependent permeability considerations;A Dahan;Molecular Pharmaceutics,2010
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