Piperidine-renin inhibitors compounds with improved physicochemical properties-Reference-Cited by-同舟云学术

Piperidine-renin inhibitors compounds with improved physicochemical properties

Published:1999-05 Issue:10 Volume:9 Page:1403-1408
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Güller Rolf,Binggeli Alfred,Breu Volker,Bur Daniel,Fischli Walter,Hirth Georges,Jenny Christian,Kansy Manfred,Montavon François,Müller Marcel,Oefner Christian,Stadler Heinz,Vieira Eric,Wilhelm Maurice,Wostl Wolfgang,Märki Hans Peter

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference17 articles.

1. Substituted piperidines - highly potent renin inhibitors due to induced fit adaptation of the active site

2. A new method for the detritylation of alcohols bearing other reducible and acid-hydrolyzable functionalities.

3. The Preparation and Some Reactions of 1-Methyl-4-phenyl-3,4-epoxypiperidine

4. Nucleophilic opening of the oxirane ring of 1-methyl-4-phenyl-3,4-epoxypiperidine

5. Coupling of Arylboronic Acids with a Partially Reduced Pyridine Derivative

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