Non-Peptide αvβ3 Antagonists. Part 4: Potent and Orally Bioavailable Chain-Shortened RGD Mimetics-Reference-Cited by-同舟云学术

Non-Peptide αvβ3 Antagonists. Part 4: Potent and Orally Bioavailable Chain-Shortened RGD Mimetics

Published:2002-09 Issue:17 Volume:12 Page:2463-2465
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Coleman Paul J.,Askew Ben C.,Hutchinson John H.,Whitman David B.,Perkins James J.,Hartman George D.,Rodan Gideon A.,Leu Chih-Tai,Prueksaritanont Thomayant,Fernandez-Metzler Carmen,Merkle Kara M.,Lynch Robert,Lynch Joseph J.,Rodan Sevgi B.,Duggan Mark E.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference17 articles.

1. New Concepts in the Pathogenesis and Treatment of Osteoporosis

2. Treatment of Postmenopausal Osteoporosis

3. Integrin-mediated signaling in the regulation of osteoclast adhesion and activation

4. Identification and in vivo efficacy of small-molecule antagonists of integrin αvβ3 (the vitronectin receptor)

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