5,5-Trans lactone-containing inhibitors of serine proteases: Identification of a novel, acylating thrombin inhibitor-Reference-Cited by-同舟云学术

5,5-Trans lactone-containing inhibitors of serine proteases: Identification of a novel, acylating thrombin inhibitor

Published:1998-11 Issue:21 Volume:8 Page:2955-2960
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Finch Harry,Pegg Neil A.,McLaren Jessica,Lowdon Andrew,Bolton Richard,Coote Steve J.,Dyer Ulrich,Montana John G.,Owen Martin R.,Dowle Mike,Buckley Doreen,Ross Barry C.,Campbell Callum,Dix Clive,Mooney Christopher,Man-Tang Chi,Patel Champa

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference31 articles.

1. Proteinase Inhibitors;Barrett,1986

2. Synthetic low-molecular weight thrombin inhibitors: molecular design and pharmacological profile

3. Orally Active .beta.-Lactam Inhibitors of Human Leukocyte Elastase. 3. Stereospecific Synthesis and Structure-Activity Relationships for 3,3-Dialkylazetidin-2-ones

4. Discovery of LB30057, a benzamidrazone-based selective oral thrombin inhibitor

Cited by 18 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Bioactive triterpenoids from Lantana camara showing anti-inflammatory activities in vitro and in vivo;Bioorganic Chemistry;2020-08

2. DBU-Promoted Cascade Annulation of Nitroarylcyclopropane-1,1-dicarbonitriles and 3-Aryl-2-cyanoacrylates: An Access to Highly Functionalized Cyclopenta[b]furan Derivatives;The Journal of Organic Chemistry;2018-11-07

3. ChemInform Abstract: 5,5-trans-Lactone-Containing Inhibitors of Serine Proteases: Identification of a Novel, Acylating Thrombin Inhibitor.;ChemInform;2010-06-17

4. N-substituted bis-C-alkyloxadiazolones as dual effectors: Efficient intermediates to amidoximes or amidines and prodrug candidates of potent antimalarials;Bioorganic & Medicinal Chemistry Letters;2009-09

5. Natural Occurring Polyphenols as Template for Drug Design. Focus on Serine Proteases;Chemical Biology & Drug Design;2009-07