Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-Positive antibacterial activity-Reference-Cited by-同舟云学术

Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-Positive antibacterial activity

Published:2003-02 Issue:4 Volume:13 Page:665-668
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Jarvest Richard L,Berge John M,Brown Murray J,Brown Pamela,Elder John S,Forrest Andrew K,Houge-Frydrych C.S.V,O'Hanlon Peter J,McNair David J,Rittenhouse Stephen,Sheppard Robert J

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference6 articles.

1. Spread of Staphylococcus aureus in Hospitals: Causes and Prevention

2. Clinical Prevalence, Antimicrobial Susceptibility, and Geographic Resistance Patterns of Enterococci: Results from the SENTRY Antimicrobial Surveillance Program, 1997–1999

3. Nanomolar Inhibitors of Staphylococcus aureus Methionyl tRNA Synthetase with Potent Antibacterial Activity against Gram-Positive Pathogens

4. Some Friedel-Crafts reactions of γ-butyrolactone

5. Reactions of Aryl Ketones and Coumarins with Iodine(III) Tris(trifluoroacetate)

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